SCHEMBL5763530

SCHEMBL5763530

COc1c(Br)ccc2c1CCC(C(=O)C(F)(F)F)NC2

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
NQO2 P16083 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
HTR2A P28223 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5732466 0.79 MTNR1A (0.47) CYP1A2MTNR1AMTNR1B
SCHEMBL5732501 0.75 DRD2 (0.33)
SCHEMBL5764333 0.73 DRD2 (0.30)
SCHEMBL5732147 0.72 SCN3A (0.30)
SCHEMBL5752287 0.70 PNMT (0.42) CYP1A2MTNR1AMTNR1B
SCHEMBL507676 0.68 ESR1 (0.52) MTNR1B
SCHEMBL3828896 0.68 BRD4 (0.36)
SCHEMBL3832960 0.68 PNMT (0.46)
SCHEMBL506348 0.67 NMT1 (0.36)
SCHEMBL5770327 0.63 MEN1 (0.40) NQO2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed