SCHEMBL5764607

SCHEMBL5764607

COCCOc1ccc2c(c1)ncn2-c1ccc2cc(-c3ccc(CN4CCOCC4)cc3)ccc2n1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FGFR1 P11362 3/20 0.47
SRC P12931 3/20 0.47
PDE2A O00408 4/20 0.44
MCHR1 Q99705 1/20 0.42
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
IKZF3 Q9UKT9 1/20 0.41
TLR7 Q9NYK1 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PDE10A Q9Y233 1/20 0.39
MAOA P21397 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ATM Q13315 1/20 0.38
KDR P35968 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
PDE11A Q9HCR9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5764733 0.92 KDR (0.45) FGFR1SRCMCHR1TLR7HRH3
SCHEMBL5767666 0.91 CHKA (0.41) FGFR1SRCMCHR1TLR7HRH3
SCHEMBL5767801 0.89 NTRK1 (0.44) FGFR1SRCTLR7MAOAATM
SCHEMBL5766984 0.87 NTRK1 (0.38) FGFR1SRCKDR
SCHEMBL5765955 0.87 LTA4H (0.36) FGFR1SRCKDR
SCHEMBL5765675 0.87 NTRK1 (0.38) FGFR1SRCKDR
SCHEMBL5764600 0.86 JAK2 (0.47) FGFR1SRCPDE2ADDB1CRBN
SCHEMBL5768958 0.85 LTA4H (0.39) FGFR1PDE2AMCHR1HRH3KDR
SCHEMBL5767363 0.85 LTA4H (0.39) FGFR1PDE2AMCHR1HRH3KDR
SCHEMBL5767404 0.84 FGFR1 (0.42) FGFR1SRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1235825-B1 NOVEL BENZOIMIDAZOLE DERIVATIVES USEFUL AS ANTIPROLIFERATIVE AGENTS PFIZER PROD INC (US) 2006-01-25 EP claimed