SCHEMBL5765100

SCHEMBL5765100

CCc1nc2ccc3c(c2nc1CC)OC(Cc1cc(C)ccc1S(=O)(=O)O)CO3

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.35
GRM1 Q13255 1/20 0.33
MAPT P10636 2/20 0.32
ALDH1A1 P00352 1/20 0.32
HTR1A P08908 3/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5768634 0.90 CA2 (0.36) CA2GRM1HTR1AGAAHSD17B10
SCHEMBL5767727 0.84 CA2 (0.36) CA2GAAHSD17B10
SCHEMBL6630732 0.83 HTR1A (0.46) CA2HTR1AGAAHSD17B10
SCHEMBL6109572 0.83 HTR1A (0.46) CA2HTR1AGAAHSD17B10
SCHEMBL6630209 0.83 HTR1A (0.37) CA2GRM1ALDH1A1HTR1A
SCHEMBL4821516 0.81 CA2 (0.38) CA2MAPTALDH1A1HTR1AHSD17B10
SCHEMBL6630585 0.80 HTR1A (0.39) CA2ALDH1A1HTR1A
SCHEMBL4335129 0.79 NR3C1 (0.37) CA2ALDH1A1HTR1AGAAHSD17B10
SCHEMBL7236260 0.78 CA2 (0.35) CA2HTR1A
SCHEMBL7240006 0.78 CA2 (0.35) CA2HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1381614-B1 ANTIDEPRESSANT AZAHETEROCYCLYLMETHYL DERIVATIVES OF 2,3-DIHYDRO-1,4-DIOXINO¬2,3-f|QUINOXALINE WYETH CORP (US) 2006-08-02 EP claimed