SCHEMBL5765610

SCHEMBL5765610

O=C(O)c1ccc2c(c1)OC=CC2

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
MAPK1 P28482 2/20 0.47
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
CA4 P22748 2/20 0.41
CA9 Q16790 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
TDP2 O95551 1/20 0.41
SRD5A2 P31213 5/20 0.40
RXRA P19793 1/20 0.38
KDM4E B2RXH2 3/20 0.37
MAPT P10636 3/20 0.37
POLB P06746 2/20 0.37
GAA P10253 1/20 0.37
CA6 P23280 1/20 0.37
PTGS2 P35354 1/20 0.37
CA7 P43166 1/20 0.37
CA14 Q9ULX7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5395777 0.86 TDP1 (0.47) ALDH1A1MAPK1CA12CA1CA2
SCHEMBL6649924 0.85 TSHR (0.49) ALDH1A1TDP2KDM4ETSHRKMT2A
SCHEMBL4538107 0.77 CA12 (0.48) ALDH1A1MAPK1CA12CA1CA2
SCHEMBL276962 0.76
SCHEMBL26654176 0.76 ALDH1A1 (0.44) ALDH1A1MAPK1CA12CA1CA2
SCHEMBL7143494 0.76 CA2 (0.40) ALDH1A1CA2KDM4EMAPTPOLB
3-Aminobenzoic Acid SCHEMBL7682790 0.75 PBRM1 (0.45) ALDH1A1CA12CA1CA2CA9
SCHEMBL547264 0.74 ESR2 (0.46) ALDH1A1MAPK1CA2KDM4EMAPT
SCHEMBL9309297 0.74 ALDH1A1 (0.57) ALDH1A1MAPK1CA12CA1CA2
SCHEMBL11296298 0.74 ALDH1A1 (0.59) ALDH1A1MAPK1CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1196692-C Substituted benzopyran derivatives for the treatment of inflammation SEARLE & CO (US) 2005-04-13 CN claimed
CN-1515566-A Substituted chromene derivative for curing inflammation G.D. 2004-07-28 CN claimed
CN-1257489-A Substituted benzopyran derivatives for the treatment of inflammation SEARLE & CO (US) 2000-06-21 CN claimed
EP-3227271-A2 HETEROCYCLIC DERIVATIVES AND USE THEREOF C&C Research Laboratories (KR) 2017-10-11 EP disclosed
CN-107001345-A Hete rocyclic derivatives and application thereof 株式会社C&C新药研究所 2017-08-01 CN disclosed
CN-1768050-A Benzopyran compounds for the treatment of inflammation PHARMACIA CORP (US) 2006-05-03 CN disclosed
EP-1631562-A1 CHROMENE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS Pharmacia Corporation (US) 2006-03-08 EP disclosed
WO-2004087687-A1 CHROMENE DERIVATIVES AS ANTI-INFLAMMATORY AGENTS PHARMACIA CORPORATION (US) 2004-10-14 WO disclosed
EP-1274700-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS Pharmacia Corporation (US) 2003-01-15 EP disclosed
WO-2001049675-A1 DIHYDROBENZOPYRANS, DIHYDROBENZOTHIOPYRANS, AND TETRAHYDROQUINOLINES FOR THE TREATMENT OF COX-2-MEDIATED DISORDERS PHARMACIA CORPORATION (US) 2001-07-12 WO disclosed