SCHEMBL5767284

SCHEMBL5767284

COc1cc2ncnc(Nc3nc4ccc(-c5cc(C(N)=O)ccc5OC)cc4s3)c2cc1OC

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 10/20 0.47
EGFR P00533 9/20 0.47
AURKB Q96GD4 5/20 0.47
AURKA O14965 3/20 0.47
BRAF P15056 2/20 0.47
RAF1 P04049 1/20 0.47
ABCG2 Q9UNQ0 2/20 0.46
CLK1 P49759 1/20 0.46
LCK P06239 1/20 0.45
TEK Q02763 1/20 0.45
RET P07949 1/20 0.43
KIF5B P33176 1/20 0.43
ABL1 P00519 1/20 0.43
DYRK1A Q13627 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5768564 0.93 EGFR (0.48) KDREGFRAURKBAURKABRAF
SCHEMBL5769764 0.87 BRAF (0.51) KDREGFRAURKBAURKABRAF
SCHEMBL5765096 0.85 KDR (0.48) KDREGFRAURKBAURKABRAF
SCHEMBL4590506 0.78 KDR (0.60) KDREGFRAURKBAURKAABCG2
SCHEMBL3949732 0.77 KDR (0.72) KDREGFRAURKBAURKA
SCHEMBL3949424 0.77 KDR (0.61) KDREGFRAURKBAURKALCK
SCHEMBL3949215 0.76 KDR (0.60) KDREGFRAURKBAURKA
SCHEMBL3947988 0.76 AURKB (0.71) KDREGFRAURKBAURKA
SCHEMBL3949004 0.75 KDR (0.73) KDREGFRAURKBAURKA
SCHEMBL3953271 0.75 KDR (0.73) KDREGFRAURKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1674467-A1 2,5- and 2,6-disubstituted benzazole derivatives useful as protein kinase inhibitors 4SC AG (DE) 2006-06-28 EP disclosed