SCHEMBL5765096

SCHEMBL5765096

COc1cc2ncnc(Nc3nc4ccc(-c5cc(C)ccc5C(N)=O)cc4s3)c2cc1OC

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDR P35968 14/20 0.48
EGFR P00533 13/20 0.47
AURKB Q96GD4 5/20 0.47
AURKA O14965 3/20 0.47
TEK Q02763 1/20 0.47
BRAF P15056 1/20 0.44
EPHA2 P29317 1/20 0.43
EPHB4 P54760 1/20 0.43
CLK1 P49759 1/20 0.42
ABCG2 Q9UNQ0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5769764 0.89 BRAF (0.51) KDREGFRAURKBAURKATEK
SCHEMBL5767284 0.85 KDR (0.47) KDREGFRAURKBAURKATEK
SCHEMBL5768564 0.85 EGFR (0.48) KDREGFRAURKBAURKATEK
SCHEMBL4590506 0.77 KDR (0.60) KDREGFRAURKBAURKACLK1
SCHEMBL3949732 0.77 KDR (0.72) KDREGFRAURKBAURKA
SCHEMBL3945407 0.77 KDR (0.54) KDREGFR
SCHEMBL3954129 0.75 KDR (0.72) KDREGFRAURKBAURKA
SCHEMBL5766719 0.75 EGFR (0.67) KDREGFRAURKBAURKATEK
SCHEMBL1505089 0.73 KDR (0.56) KDREGFRCLK1ABCG2
SCHEMBL3947263 0.73 KDR (0.72) KDREGFRAURKBAURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1674467-A1 2,5- and 2,6-disubstituted benzazole derivatives useful as protein kinase inhibitors 4SC AG (DE) 2006-06-28 EP disclosed