SCHEMBL5770352

SCHEMBL5770352

CNCCCOc1cccc2c3ccccc3n(C)c12

nearest known ligand 0.58

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 3/20 0.58
SLC6A4 P31645 2/20 0.58
HTR1B P28222 7/20 0.52
HTR1D P28221 1/20 0.52
ALKBH5 Q6P6C2 1/20 0.46
FTO Q9C0B1 1/20 0.46
HTR6 P50406 1/20 0.44
TP53 P04637 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
KCNA3 P22001 1/20 0.42
LMNA P02545 1/20 0.42
NR2E1 Q9Y466 1/20 0.42
MCL1 Q07820 1/20 0.41
GPR3 P46089 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5749824 0.96 HTR1B (0.57) HRH1SLC6A4HTR1BHTR1DALKBH5
SCHEMBL5747747 0.88 HTR1B (0.56) HRH1SLC6A4HTR1BHTR1DALKBH5
SCHEMBL5747639 0.86 HTR1B (0.61) HRH1SLC6A4HTR1BHTR1DALKBH5
SCHEMBL5771872 0.84 HTR1B (0.60) HRH1SLC6A4HTR1BHTR1DALKBH5
SCHEMBL5747516 0.83 HTR1B (0.54) HTR1BALKBH5FTOKCNA3LMNA
SCHEMBL5748798 0.81 HTR1B (0.53) HTR1BALKBH5FTOHTR6TP53
SCHEMBL15466278 0.79 ALKBH5 (0.54) ALKBH5FTOTP53L3MBTL1LMNA
SCHEMBL5748074 0.79 SLC6A4 (0.53) HRH1SLC6A4HTR1BHTR1DHTR6
SCHEMBL5748094 0.78 CYP2D6 (0.55) HRH1HTR6CYP1A2L3MBTL1
SCHEMBL5748021 0.77 HTR1B (0.50) HRH1SLC6A4HTR1BHTR1DALKBH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed