SCHEMBL5747747

SCHEMBL5747747

CCNCCCOc1cccc2c3ccccc3n(C)c12

nearest known ligand 0.56

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 4/20 0.56
ADRB2 P07550 2/20 0.46
ALKBH5 Q6P6C2 1/20 0.45
FTO Q9C0B1 1/20 0.45
SLC6A4 P31645 4/20 0.43
HRH1 P35367 1/20 0.43
KMT2A Q03164 1/20 0.42
HTR1D P28221 1/20 0.41
KCNA3 P22001 1/20 0.41
NR2E1 Q9Y466 1/20 0.41
HTR1A P08908 2/20 0.40
MCL1 Q07820 1/20 0.40
GPR3 P46089 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5747639 0.96 HTR1B (0.61) HTR1BADRB2ALKBH5FTOSLC6A4
SCHEMBL5771872 0.88 HTR1B (0.60) HTR1BADRB2ALKBH5FTOSLC6A4
SCHEMBL5770352 0.88 HRH1 (0.58) HTR1BALKBH5FTOSLC6A4HRH1
SCHEMBL5749824 0.86 HTR1B (0.57) HTR1BALKBH5FTOSLC6A4HRH1
SCHEMBL5747516 0.82 HTR1B (0.54) HTR1BALKBH5FTOKMT2AKCNA3
SCHEMBL15466278 0.81 ALKBH5 (0.54) ALKBH5FTOKMT2AGPR3
SCHEMBL5748798 0.80 HTR1B (0.53) HTR1BALKBH5FTOKMT2AKCNA3
SCHEMBL5746733 0.80 HTR1B (0.51) HTR1BADRB2SLC6A4HRH1KCNA3
SCHEMBL5745853 0.79 HTR1B (0.53) HTR1BADRB2SLC6A4HRH1KMT2A
SCHEMBL5748021 0.78 HTR1B (0.50) HTR1BALKBH5FTOSLC6A4HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1711463-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2006-10-18 EP disclosed
WO-2005077899-A2 AMINO-SUBSTITUTED TRICYCLIC DERIVATIVES AND METHODS OF USE ABBOTT LABORATORIES (US) 2005-08-25 WO disclosed