SCHEMBL5771242

SCHEMBL5771242

COc1ccc(S(=O)(=O)C(N)(CC(C)(C)CCCN)[C@H](O)[C@H](Cc2ccccc2)NC(=O)Oc2ccoc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 4/20 0.38
MMP2 P08253 2/20 0.38
MMP3 P08254 2/20 0.38
PDE4A P27815 2/20 0.38
PDE4B Q07343 2/20 0.38
PDE4C Q08493 2/20 0.38
PDE4D Q08499 2/20 0.38
MMP9 P14780 2/20 0.36
MMP13 P45452 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5771964 0.96 MMP1 (0.38) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL5771248 0.83 MMP9 (0.40) MMP1MMP2MMP3MMP9MMP13
SCHEMBL5772323 0.79 ABCB1 (0.52)
SCHEMBL5771716 0.79 ABCB1 (0.52)
SCHEMBL5770232 0.79 MLNR (0.44)
SCHEMBL5770234 0.79 MLNR (0.44)
SCHEMBL5770237 0.79 MMP2 (0.41) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL5771246 0.76 MMP1 (0.42) MMP1MMP2MMP3PDE4APDE4B
SCHEMBL5773479 0.75 ABCB1 (0.54)
SCHEMBL5773722 0.75 ABCB1 (0.54)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed