SCHEMBL5771660

SCHEMBL5771660

CC1CC(c2ncc3nccc-3[nH]2)CC(c2cccc(Cl)c2)N1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SLC9A1 P19634 1/20 0.32
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
ADRA1A P35348 1/20 0.31
TRPM4 Q8TD43 1/20 0.31
TRPM5 Q9NZQ8 1/20 0.31
NPY5R Q15761 1/20 0.30
GSK3B P49841 1/20 0.30
SCN2A Q99250 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5775581 0.98 SLC9A1 (0.31) SLC9A1KDM1AMAOB
SCHEMBL5771458 0.88 HDAC4 (0.32) GSK3B
SCHEMBL5772547 0.87 MAPT (0.32) KDM1AMAOB
SCHEMBL5771433 0.86 NPY5R (0.32) NPY5R
Hydrochloric Acid SCHEMBL5772584 0.86 MAPT (0.32) KDM1AMAOB
Hydrochloric Acid SCHEMBL5775499 0.86 HPGDS (0.32)
Hydrochloric Acid SCHEMBL5774750 0.86 HDAC4 (0.31) GSK3B
Hydrochloric Acid SCHEMBL5775416 0.84 NPY5R (0.31) NPY5R
SCHEMBL5773116 0.84
SCHEMBL5770939 0.83 CYP2D6 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed