SCHEMBL5772158

SCHEMBL5772158

CC(C)(CCCCO)C(NC[C@@H](O)[C@H](Cc1ccccc1)NC(=O)O)S(=O)(=O)c1ccc2c(c1)OCO2

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 10/20 0.38
CTSD P07339 1/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
ADRB3 P13945 1/20 0.37
VIPR2 P41587 1/20 0.37
ITGB3 P05106 1/20 0.36
ITGAV P06756 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.35
MEN1 O00255 1/20 0.35
MAPT P10636 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6763344 0.92 BACE1 (0.39) BACE1CTSD
SCHEMBL7392821 0.81 CTSD (0.49) BACE1CTSD
SCHEMBL1601744 0.80 SPPL2A (0.42) CTSDMAPT
SCHEMBL1601742 0.80 SPPL2A (0.42) CTSDMAPT
SCHEMBL6051065 0.77 MAOB (0.42) CTSD
SCHEMBL4347480 0.77 MAOA (0.44) BACE1CTSDMAPT
SCHEMBL6915284 0.74 MAOB (0.40) BACE1CTSDBACE2
SCHEMBL5771630 0.74 MEP1B (0.39) BACE1CTSDMAPTSMN1; SMN2
SCHEMBL4352403 0.74 ABCB1 (0.39) BACE1MAPTSMN1; SMN2
SCHEMBL8898130 0.73 BACE1 (0.39) BACE1CTSDBACE2ADRB3VIPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed