SCHEMBL5772805

SCHEMBL5772805

Cc1nc(N2CC=CC2)c2nc(-c3ccc(Cl)c(Cl)c3)cc-2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.39
NPY5R Q15761 4/20 0.39
KMO O15229 2/20 0.36
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
ADORA3 P0DMS8 2/20 0.34
ADORA1 P30542 1/20 0.34
AR P10275 1/20 0.34
PIK3CA P42336 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 2/20 0.33
PIM1 P11309 1/20 0.33
TYMP P19971 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5778150 0.98 HRH4 (0.38) HRH4NPY5RKMOKDM4ENPC1
SCHEMBL5772845 0.86 NPY5R (0.41) NPY5RNPC1RAB9AADORA3ADORA1
Hydrochloric Acid SCHEMBL5777029 0.84 NPY5R (0.40) NPY5RNPC1RAB9AADORA3ADORA1
SCHEMBL5773685 0.83 NPY5R (0.40) HRH4NPY5RKDM4EMAPTALDH1A1
Hydrochloric Acid SCHEMBL5773424 0.81 NPY5R (0.39) HRH4NPY5RKDM4EMAPTALDH1A1
SCHEMBL5772572 0.79 KMO (0.43) NPY5RKMONPC1RAB9AKMT2A
SCHEMBL5772107 0.78 XDH (0.43) NPY5RKDM4EARALDH1A1HPGD
SCHEMBL5775574 0.77 KMO (0.44) NPY5RKMOKDM4ENPC1RAB9A
Hydrochloric Acid SCHEMBL5774382 0.77 XDH (0.41) NPY5RKDM4EARALDH1A1HPGD
SCHEMBL5775406 0.76 NPY5R (0.56) NPY5RKDM4ERAB9AADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed