SCHEMBL5773246

SCHEMBL5773246

CCCc1nc(C2CCNC(c3ccccc3)C2)c2nccc-2[nH]1

nearest known ligand 0.34

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 1/20 0.34
ADORA3 P0DMS8 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5772701 0.98 CHRNA7 (0.33) CHRNA7ADORA3ADORA2AADORA1
SCHEMBL5771094 0.89 PARP1 (0.31)
Hydrochloric Acid SCHEMBL7182724 0.88 PARP1 (0.30)
SCHEMBL5774419 0.83 PTPN11 (0.30)
SCHEMBL7959871 0.83 KDM4E (0.35) CHRNA7
Hydrochloric Acid SCHEMBL5773960 0.82 KDM4E (0.34) CHRNA7
Hydrochloric Acid SCHEMBL5774721 0.82
SCHEMBL5776304 0.81 PRCP (0.32)
Hydrochloric Acid SCHEMBL5775502 0.80 NOS1 (0.34)
Hydrochloric Acid SCHEMBL5775517 0.80 MMP12 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed