SCHEMBL5773890

SCHEMBL5773890

Cc1nc(C2CCNCC2)c2sc(C(C)(C)C)cc2n1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRM4 P08173 1/20 0.38
KIT P10721 1/20 0.38
PDPK1 O15530 1/20 0.36
NPY5R Q15761 1/20 0.35
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TLR9 Q9NR96 2/20 0.32
TLR8 Q9NR97 2/20 0.32
TLR7 Q9NYK1 2/20 0.32
NMT1 P30419 2/20 0.31
SOS1 Q07889 3/20 0.31
KCNH2 Q12809 1/20 0.31
HTR2C P28335 2/20 0.31
PRKCI P41743 1/20 0.30
HRH4 Q9H3N8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7188454 0.99 CHRM4 (0.37) CHRM4KITPDPK1NPY5RMEN1
SCHEMBL5773747 0.76 NPY5R (0.51) CHRM4KITNPY5RMEN1KMT2A
Hydrochloric Acid SCHEMBL5774370 0.75 NPY5R (0.50) KITNPY5RMEN1KMT2ANPC1
SCHEMBL5771159 0.74 RAB9A (0.42) CHRM4KITNPY5RNPC1RAB9A
SCHEMBL5772338 0.74 KCNH2 (0.42) KITPDPK1NPY5RRAB9AKCNH2
Hydrochloric Acid SCHEMBL5773821 0.73 RAB9A (0.44) CHRM4KITNPY5RNPC1RAB9A
SCHEMBL19198488 0.73 MEN1 (0.40) CHRM4PDPK1NPY5RMEN1KMT2A
Hydrochloric Acid SCHEMBL5773172 0.72 KCNH2 (0.41) KITPDPK1NPY5RRAB9AKCNH2
SCHEMBL12105218 0.72 PDPK1 (0.42) PDPK1MEN1KMT2ANMT1PRKCI
SCHEMBL5772009 0.65 MEN1 (0.67) NPY5RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6583154-B1 Neuropeptide Y antagonist; pyrrolo-(3,2-b)pyridines and pyrrolo-(3,2-d)pyrimidines AMGEN INC. 2003-06-24 US disclosed