SCHEMBL5772338

SCHEMBL5772338

Cc1nc(C2CCNCC2)c2sc(-c3ccc(F)cc3)cc2n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 4/20 0.42
RAB9A P51151 1/20 0.41
KIT P10721 2/20 0.41
MKNK1 Q9BUB5 1/20 0.41
MKNK2 Q9HBH9 1/20 0.41
SLC6A2 P23975 1/20 0.40
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
TYK2 P29597 1/20 0.40
PDPK1 O15530 1/20 0.40
MAPK11 Q15759 2/20 0.39
MAPK14 Q16539 2/20 0.39
MAPK13 O15264 1/20 0.39
RAF1 P04049 1/20 0.39
MAPK9 P45984 1/20 0.39
MAPK12 P53778 1/20 0.39
NPY5R Q15761 1/20 0.39
ACHE P22303 1/20 0.37
PRKCI P41743 1/20 0.36
CDC7 O00311 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5773172 0.98 KCNH2 (0.41) KCNH2RAB9AKITMKNK1MKNK2
SCHEMBL5771159 0.88 RAB9A (0.42) KCNH2RAB9AKITNPY5RPRKCI
SCHEMBL5773747 0.88 NPY5R (0.51) KCNH2RAB9AKITNPY5RPRKCI
Hydrochloric Acid SCHEMBL5773821 0.87 RAB9A (0.44) KCNH2RAB9AKITNPY5RPRKCI
Hydrochloric Acid SCHEMBL5774370 0.87 NPY5R (0.50) KCNH2RAB9AKITNPY5RPRKCI
SCHEMBL5773890 0.74 CHRM4 (0.38) KCNH2RAB9AKITPDPK1NPY5R
Hydrochloric Acid SCHEMBL7188454 0.73 CHRM4 (0.37) KCNH2RAB9AKITPDPK1NPY5R
SCHEMBL5772334 0.69 NPY5R (0.78) KCNH2NPY5RPRKCI
Hydrochloric Acid SCHEMBL5773169 0.67 NPY5R (0.74) KCNH2KITNPY5RPRKCI
SCHEMBL5776584 0.66 NPY5R (0.47) RAB9ANPY5RPRKCICDC7DBF4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed