SCHEMBL5774465

SCHEMBL5774465

COc1c(F)cc(F)cc1C(C)(C)CC(O)(C=O)C(F)(F)F.COc1c(F)cc(F)cc1C(C)(C)CC(O)(CNc1cccc2[nH]ncc12)C(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 12/20 0.46
PGR P06401 7/20 0.46
NR3C2 P08235 4/20 0.37
TRPV1 Q8NER1 5/20 0.36
NPC1 O15118 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
HPGD P15428 1/20 0.35
CYP2C19 P33261 1/20 0.35
HTT P42858 1/20 0.35
RAB9A P51151 1/20 0.35
DHPS P49366 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5797178 0.93 NR3C1 (0.51) NR3C1PGRNR3C2TRPV1
SCHEMBL5779425 0.87 NR3C1 (0.43) NR3C1PGRTRPV1DHPS
SCHEMBL6403409 0.84 NR3C1 (0.50) NR3C1PGRNR3C2TRPV1NPC1
SCHEMBL5774468 0.84 TRPV1 (0.33) NR3C1PGRNR3C2TRPV1NPC1
SCHEMBL5779746 0.83 NR3C1 (0.41) NR3C1PGRNR3C2TRPV1DHPS
SCHEMBL6408601 0.82 NR3C1 (0.53) NR3C1PGRNR3C2TRPV1NPC1
SCHEMBL5778544 0.81 NR3C1 (0.68) NR3C1PGRNR3C2
SCHEMBL4732633 0.80 NR3C1 (0.57) NR3C1PGRNR3C2TRPV1NPC1
SCHEMBL6405053 0.80 NR3C1 (0.55) NR3C1PGRNR3C2
SCHEMBL5780477 0.79 NR3C1 (0.60) NR3C1PGRNR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1638945-A1 HETEROCYCLICALLY SUBSTITUTED PENTANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS Schering Aktiengesellschaft (DE) 2006-03-29 EP disclosed
WO-2005003098-A1 HETEROCYCLICALLY SUBSTITUTED PENTANOL DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF, AND USE THEREOF AS ANTI-INFLAMMATORY AGENTS SCHERING AKTIENGESELLSCHAFT (DE) 2005-01-13 WO disclosed