SCHEMBL5774467

SCHEMBL5774467

Cc1nc(C2CCNCC2)c2nc(-c3cc(F)cc(F)c3)c(C)c-2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TLR9 Q9NR96 13/20 0.37
TLR8 Q9NR97 13/20 0.37
TLR7 Q9NYK1 13/20 0.37
TNKS O95271 4/20 0.36
TNKS2 Q9H2K2 4/20 0.36
PARP1 P09874 2/20 0.36
KCNH2 Q12809 2/20 0.36
MAPK13 O15264 1/20 0.36
RAF1 P04049 1/20 0.36
MAPK9 P45984 1/20 0.36
MAPK12 P53778 1/20 0.36
MAPK11 Q15759 1/20 0.36
MAPK14 Q16539 1/20 0.36
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774851 0.88 MAPK14 (0.48) TNKSTNKS2PARP1KCNH2MAPK13
Hydrochloric Acid SCHEMBL5773943 0.84 MAPK14 (0.42) TLR9TLR8TLR7TNKSTNKS2
SCHEMBL5775115 0.81 USP7 (0.41) TLR9TLR8TLR7MAPK13RAF1
Hydrochloric Acid SCHEMBL5775248 0.81 KDM4E (0.44) KCNH2
SCHEMBL7960972 0.80 SLC6A2 (0.37) TLR9TLR8TLR7MAPK13MAPK9
SCHEMBL8125046 0.79 MEN1 (0.44) TLR9TLR7
SCHEMBL5776541 0.75 MAPK14 (0.45) TLR9TLR8TLR7TNKSTNKS2
Hydrochloric Acid SCHEMBL5807137 0.75 KDM4E (0.43) TLR9TLR8TLR7KCNH2MAPK13
SCHEMBL5774480 0.71 KDM4E (0.44) TLR9TLR8TLR7KCNH2MAPK13
Hydrochloric Acid SCHEMBL5773701 0.70 KDM4E (0.47) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed