SCHEMBL5774977

SCHEMBL5774977

COc1ccc(S(=O)(=O)N(Cc2ccccc2)[C@H](NC(=O)Oc2coc3occc23)[C@@H](C)O)cc1CC(C)(C)CCN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.32
KMT2A Q03164 2/20 0.32
ACHE P22303 2/20 0.31
HTT P42858 2/20 0.31
TAS2R14 Q9NYV8 2/20 0.31
BCHE P06276 1/20 0.31
BMP1 P13497 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5774835 0.89 HTT (0.30) KMT2AHTT
SCHEMBL5771487 0.87 KMT2A (0.33) L3MBTL1KMT2AACHEHTTTAS2R14
SCHEMBL6199940 0.85 PSEN1 (0.38) L3MBTL1KMT2AHTT
SCHEMBL1602478 0.85 ALDH1A1 (0.38) L3MBTL1KMT2AHTTTAS2R14MEN1
SCHEMBL6621241 0.81 PDE4B (0.44)
SCHEMBL1602317 0.77 ABCB1 (0.47)
SCHEMBL1600923 0.77 ABCB1 (0.47)
SCHEMBL1601957 0.77 TP53 (0.39) KMT2AHTTTAS2R14ALDH1A1GAA
SCHEMBL1602845 0.75 KMT2A (0.38) KMT2AHTTTAS2R14ALDH1A1
SCHEMBL1602738 0.75 BMP1 (0.38) KMT2AHTTTAS2R14BMP1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed