SCHEMBL5771487

SCHEMBL5771487

COc1ccc(S(=O)(=O)N(Cc2ccccc2)[C@H](NC(=O)Oc2ccoc2)[C@@H](C)O)cc1CC(C)(C)CCN(Cc1ccccc1)Cc1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.33
CASP1 P29466 1/20 0.33
CASP3 P42574 1/20 0.33
CASP7 P55210 1/20 0.33
CASP8 Q14790 1/20 0.33
BMP1 P13497 3/20 0.33
TAS2R14 Q9NYV8 2/20 0.33
MMP2 P08253 2/20 0.33
MMP9 P14780 2/20 0.33
ACHE P22303 2/20 0.33
MMP8 P22894 1/20 0.33
HTT P42858 2/20 0.32
BCHE P06276 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6199940 0.87 PSEN1 (0.38) KMT2AMMP2MMP9MMP8HTT
SCHEMBL1602478 0.87 ALDH1A1 (0.38) KMT2ATAS2R14MMP2MMP9MMP8
SCHEMBL5774977 0.87 L3MBTL1 (0.32) KMT2ABMP1TAS2R14ACHEHTT
SCHEMBL6617043 0.80 PDE4B (0.48)
SCHEMBL1600923 0.79 ABCB1 (0.47)
SCHEMBL1602317 0.79 ABCB1 (0.47)
SCHEMBL1601957 0.79 TP53 (0.39) KMT2ATAS2R14MMP2MMP9MMP8
SCHEMBL1602845 0.77 KMT2A (0.38) KMT2ATAS2R14MMP2MMP9MMP8
SCHEMBL1602738 0.77 BMP1 (0.38) KMT2ABMP1TAS2R14MMP2MMP9
SCHEMBL1601671 0.76 MAPT (0.36) KMT2ATAS2R14MMP2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1637518-A2 Inhibitors of aspartyl protease Vertex Pharmaceuticals Incorporated (US) 2006-03-22 EP disclosed