SCHEMBL5777601

SCHEMBL5777601

CCOC(=O)c1nc(C(C)C)ns1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.40
MAPT P10636 5/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP1A2 P05177 3/20 0.39
CYP2C19 P33261 1/20 0.36
HPGD P15428 4/20 0.36
GAA P10253 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
POLB P06746 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
HSP90AA1 P07900 1/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9029404 0.89 HTT (0.37) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL23796408 0.87 ALDH1A1 (0.39) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL23795980 0.87 CYP1A2 (0.37) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL23796111 0.81 CYP1A2 (0.33) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL22578954 0.79 CYP1A2 (0.43) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL29117128 0.76 LMNA (0.43) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL29117129 0.76 LMNA (0.43) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL25219857 0.76 CYP1A2 (0.41) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL18039508 0.76 CYP1A2 (0.41) ALDH1A1MAPTRAB9ANPC1MEN1
SCHEMBL23796030 0.75 CYP1A2 (0.40) ALDH1A1MAPTRAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed
US-5583092-A PLANT ANTIGROWTH AGENTS AMERICAN CYANAMID COMPANY (US) 1996-12-10 US disclosed
EP-0726261-A1 Herbidical 1,2,4 thiadiazoles American Cyanamid Company (US) 1996-08-14 EP disclosed
EP-0726260-A1 Herbicidal (1,2,4)thiadiazoles AMERICAN CYANAMID COMPANY (US) 1996-08-14 EP disclosed