SCHEMBL5778038

SCHEMBL5778038

Fc1cc(Br)c2c(CCc3ccc(Cl)cc3)c3n(c2c1)CC[C]3

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 7/20 0.42
PTGER1 P34995 1/20 0.32
PTGER4 P35408 1/20 0.32
PTGFR P43088 1/20 0.32
PTGER3 P43115 1/20 0.32
PTGER2 P43116 1/20 0.32
PTGIR P43119 1/20 0.32
PTGDR Q13258 1/20 0.32
PDE2A O00408 1/20 0.31
HTR1A P08908 1/20 0.31
DRD2 P14416 1/20 0.31
DRD1 P21728 1/20 0.31
DRD5 P21918 1/20 0.31
HTR2A P28223 1/20 0.31
DRD3 P35462 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
SIGMAR1 Q99720 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778034 0.80 TBXA2R (0.43) TBXA2RPTGER1PTGER4PTGFRPTGER3
SCHEMBL6727090 0.65 TBXA2R (0.75) TBXA2RPTGER1PTGER4PTGFRPTGER3
SCHEMBL2135113 0.56 TAAR1 (0.68)
SCHEMBL12147413 0.55 TAAR1 (0.50)
SCHEMBL18550393 0.55 TAAR1 (0.54) HTR2A
SCHEMBL27891098 0.54 TAAR1 (0.57) DRD2
SCHEMBL14143081 0.53 PSEN1 (0.51) HTR2A
SCHEMBL10501653 0.52 DRD2 (0.58) HTR1ADRD2DRD1DRD5HTR2A
SCHEMBL2303570 0.52 DRD2 (0.54) HTR1ADRD2DRD1DRD5HTR2A
SCHEMBL1868021 0.52 PTGS1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed