SCHEMBL5778034

SCHEMBL5778034

Fc1cc(Br)c2c(CCc3ccc(Cl)cc3)c3n(c2c1)CC[CH]3

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 8/20 0.43
DRD2 P14416 3/20 0.34
HTR1A P08908 2/20 0.34
HTR2A P28223 2/20 0.34
DRD3 P35462 2/20 0.34
TMEM97 Q5BJF2 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
DRD1 P21728 1/20 0.34
DRD5 P21918 1/20 0.34
MAPT P10636 1/20 0.33
PTGER1 P34995 1/20 0.32
PTGER4 P35408 1/20 0.32
PTGFR P43088 1/20 0.32
PTGER3 P43115 1/20 0.32
PTGER2 P43116 1/20 0.32
PTGIR P43119 1/20 0.32
PTGDR Q13258 1/20 0.32
HTR2C P28335 1/20 0.32
HRH1 P35367 1/20 0.32
PDE2A O00408 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5778038 0.80 TBXA2R (0.42) TBXA2RDRD2HTR1AHTR2ADRD3
SCHEMBL6727090 0.66 TBXA2R (0.75) TBXA2RPTGER1PTGER4PTGFRPTGER3
SCHEMBL5777733 0.65 TBXA2R (0.42) TBXA2RDRD2HTR1A
SCHEMBL6579205 0.61 PTGDR (0.55) TBXA2RDRD3MAPTPTGER1PTGER4
SCHEMBL2135113 0.57 TAAR1 (0.68) IDO1
SCHEMBL12147413 0.56 TAAR1 (0.50) IDO1
SCHEMBL18550393 0.56 TAAR1 (0.54) HTR2AIDO1
SCHEMBL27891098 0.55 TAAR1 (0.57) DRD2IDO1
SCHEMBL14143081 0.54 PSEN1 (0.51) HTR2AMAPTHTR2C
SCHEMBL10501653 0.53 DRD2 (0.58) DRD2HTR1AHTR2ADRD3TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1395590-B1 DIHYDROPYRROLO¬1,2-A|INDOLE AND TETRAHYDROPYRIDO¬1,2-A|INDOLE DERIVATIVES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS MERCK FROSST CANADA INC (CA) 2006-09-27 EP disclosed