SCHEMBL5778634

SCHEMBL5778634

CC1CCCCN1c1ncccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.48
LMNA P02545 4/20 0.48
HTT P42858 3/20 0.48
NCOA3 Q9Y6Q9 1/20 0.48
BCHE P06276 1/20 0.46
ACHE P22303 1/20 0.46
DYRK1A Q13627 1/20 0.45
ALDH1A1 P00352 3/20 0.45
GAA P10253 1/20 0.45
MEN1 O00255 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
JAK3 P52333 1/20 0.43
TSHR P16473 2/20 0.42
XBP1 P17861 1/20 0.42
ALOX15 P16050 2/20 0.42
MAPT P10636 2/20 0.42
USP2 O75604 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26691316 0.94 DYRK1A (0.49) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL5774649 0.94 DYRK1A (0.49) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL8272981 0.94 DYRK1A (0.49) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL25247899 0.86 SLC6A7 (0.42) SMN1; SMN2LMNAHTTNCOA3DYRK1A
SCHEMBL5778408 0.86 SLC6A7 (0.42) SMN1; SMN2LMNAHTTNCOA3DYRK1A
SCHEMBL17210377 0.80 ALDH1A1 (0.44) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL17201983 0.80 ALDH1A1 (0.44) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL13402936 0.80 DYRK1A (0.48) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL27268114 0.79 LMNA (0.50) SMN1; SMN2LMNAHTTNCOA3BCHE
SCHEMBL27998984 0.77 KDM4E (0.36) SMN1; SMN2LMNAHTTNCOA3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105814056-A Purine derivatives as modulators of TNF activity UCB生物制药私人有限公司 2016-07-27 CN disclosed
EP-1644358-A2 BIARYL PIPERAZINYL-PYRIDINE ANALOGUES NEUROGEN CORPORATION (US) 2006-04-12 EP disclosed
WO-2005007648-A2 BIARYL PIPERAZINYL-PYRIDINE ANALOGUES NEUROGEN CORPORATION (US) 2005-01-27 WO disclosed