SCHEMBL5778644

SCHEMBL5778644

Nc1cccc(C(=O)Nc2nc(-c3ccccc3)cs2)c1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 1/20 0.69
MAPT P10636 4/20 0.68
ALDH1A1 P00352 2/20 0.68
MEN1 O00255 1/20 0.68
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
HTT P42858 1/20 0.68
KMT2A Q03164 1/20 0.68
PARP1 P09874 1/20 0.65
LMNA P02545 1/20 0.65
RRM1 P23921 1/20 0.61
RRM2B Q7LG56 1/20 0.61
PHGDH O43175 2/20 0.60
ADORA3 P0DMS8 1/20 0.60
RAB9A P51151 2/20 0.59
NPC1 O15118 1/20 0.59
GAA P10253 1/20 0.59
NPSR1 Q6W5P4 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15688657 0.93 SCD (0.69) SCDMAPTALDH1A1MEN1CYP1A2
SCHEMBL1270375 0.87 SCD (0.89) SCDMAPTALDH1A1MEN1HTT
SCHEMBL26673963 0.86 SCD (0.74) SCDMAPTALDH1A1MEN1KMT2A
SCHEMBL2754070 0.85 ADORA3 (0.74) SCDMAPTALDH1A1MEN1CYP1A2
SCHEMBL2754003 0.85 SCD (0.69) SCDMAPTALDH1A1MEN1CYP1A2
SCHEMBL2753571 0.82 ALDH1A1 (0.85) SCDMAPTALDH1A1MEN1CYP1A2
SCHEMBL10966343 0.82 HDAC3 (0.65) MAPTALDH1A1MEN1HTTKMT2A
SCHEMBL16562127 0.82 SCD (1.00) SCDMAPTALDH1A1PARP1LMNA
SCHEMBL23674562 0.81 SCD (0.84) SCDMAPTALDH1A1MEN1HTT
SCHEMBL5774803 0.81 MEN1 (1.00) SCDMAPTALDH1A1MEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed