SCHEMBL5774803

SCHEMBL5774803

O=C(Nc1nc(-c2ccccc2)cs1)c1cccc([N+](=O)[O-])c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 1.00
KMT2A Q03164 5/20 1.00
MAPT P10636 4/20 1.00
ALDH1A1 P00352 3/20 1.00
HTT P42858 2/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
CYP2C9 P11712 1/20 1.00
CYP2C19 P33261 1/20 1.00
POLB P06746 1/20 0.82
RAB9A P51151 2/20 0.80
BAZ1A Q9NRL2 1/20 0.71
SCD O00767 1/20 0.63
CSNK2A1 P68400 3/20 0.62
TP53 P04637 1/20 0.61
GAA P10253 1/20 0.60
PARP1 P09874 1/20 0.60
ADORA3 P0DMS8 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15688998 0.93 MEN1 (0.87) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL10962764 0.83 KMT2A (0.74) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL1270375 0.83 SCD (0.89) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL27771294 0.82 KMT2A (0.77) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL10808167 0.82 BAZ1A (0.79) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL10922701 0.82 KMT2A (0.72) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL7128794 0.81 MEN1 (0.69) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL5778644 0.81 SCD (0.69) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL2754070 0.81 ADORA3 (0.74) MEN1KMT2AMAPTALDH1A1HTT
SCHEMBL2754003 0.81 SCD (0.69) MEN1KMT2AMAPTALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1652839-A2 Drug efflux pump inhibitor DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-05-03 EP disclosed
EP-1227084-B1 DRUG DISCHARGE PUMP INHIBITORS TRINE PHARMACEUTICALS INC (US) 2005-12-14 EP disclosed
EP-1227084-A1 DRUG DISCHARGE PUMP INHIBITORS Microcide Pharmaceuticals, Inc. (US) 2002-07-31 EP disclosed