SCHEMBL5778714

SCHEMBL5778714

Clc1cc(Oc2nccc3ccccc23)ncn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.48
DRD1 P21728 4/20 0.38
FFAR1 O14842 1/20 0.38
CYP2A6 P11509 1/20 0.38
F12 P00748 1/20 0.38
PLAU P00749 1/20 0.38
NCF1 P14598 1/20 0.38
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
NOS2 P35228 1/20 0.38
BACE1 P56817 1/20 0.38
LMNA P02545 2/20 0.37
MAPT P10636 2/20 0.37
CYP3A4 P08684 1/20 0.37
APEX1 P27695 1/20 0.37
MAPK1 P28482 1/20 0.37
PMP22 Q01453 1/20 0.37
KLK5 Q9Y337 1/20 0.37
EGFR P00533 2/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31498832 0.77 TRPA1 (0.60) TRPA1DRD1FFAR1CYP2A6F12
SCHEMBL6110247 0.77 TRPA1 (0.60) TRPA1DRD1FFAR1CYP2A6F12
SCHEMBL5968524 0.74 TRPV1 (0.59) NPC1RAB9ASMN1; SMN2
SCHEMBL3875440 0.73 KDR (0.42) NCF1MAPTMAPK1EGFRALDH1A1
SCHEMBL3876878 0.72 EGFR (0.38) LMNAMAPTCYP3A4MAPK1EGFR
SCHEMBL3875328 0.72 NPC1 (0.39) CYP2A6LMNAMAPTMAPK1EGFR
SCHEMBL7790214 0.72 HAO1 (0.47) CYP2A6LMNAMAPTNPC1RAB9A
SCHEMBL191210 0.71 NPC1 (0.61) MAPK1NPC1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL1093339 0.71 TRPA1 (0.54) TRPA1DRD1FFAR1CYP2A6F12
SCHEMBL26697193 0.69 ALDH1A1 (0.39) LMNAMAPTMAPK1NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720868-A1 PYRIMIDINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS AND THEIR USE IN THE TREATMENT OF PAIN AMGEN INC. (US) 2006-11-15 EP disclosed
WO-2005077944-A1 PYRIMIDINE DERIVATIVES FOR USE AS VANILLOID RECEPTOR LIGANDS AND THEIR USE IN THE TREATMENT OF PAIN AMGEN INC. (US) 2005-08-25 WO disclosed