SCHEMBL5779683

SCHEMBL5779683

CCOOC(=O)c1cn(C)c2cc(CNc3nccn3C(c3ccccc3)(c3ccccc3)c3ccccc3)ccc2c1=O

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 10/20 0.36
S1PR3 Q99500 4/20 0.36
P2RX3 P56373 1/20 0.34
KDR P35968 1/20 0.33
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
THRB P10828 1/20 0.32
CNR1 P21554 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12372084 0.92 P2RX3 (0.42) S1PR1S1PR3P2RX3KDRRAB9A
SCHEMBL4388255 0.89 S1PR1 (0.40) S1PR1S1PR3KDRPOLBNPC1
SCHEMBL7055717 0.80 S1PR1 (0.41) S1PR1S1PR3NPC1RAB9AALDH1A1
SCHEMBL5779687 0.78 NPC1 (0.34) POLBNPC1RAB9AALDH1A1TP53
SCHEMBL4654781 0.77 P2RX3 (0.40) P2RX3ALDH1A1CNR1
SCHEMBL8635242 0.76 NPC1 (0.31) KDRNPC1RAB9AALDH1A1
SCHEMBL27608112 0.76 KMT2A (0.35) ALDH1A1TP53
SCHEMBL7052174 0.76 P2RX3 (0.39) P2RX3ALDH1A1CNR1
SCHEMBL4654929 0.74 CAMK2D (0.37) CNR1
SCHEMBL12398941 0.73 P2RX3 (0.42) S1PR1S1PR3P2RX3POLBRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0944619-B1 NOVEL INTEGRIN RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB PHARMA CO (US) 2006-10-11 EP disclosed
US-6358976-B1 FOR THERAPY AND PROPHYLAXIS OF CANCER METASTASIS, DIABETIC RETINOPATHY, NEOVASCULAR GLAUCOMA, THROMBOSIS, RESTENOSIS, OSTEOPOROSIS, OR MACULAR DEGENERATION LANTHEUS MI REAL ESTATE, LLC 2002-03-19 US disclosed
US-6130231-A SUBSTITUTED 2,3-DIHYDROQUINOLIN-4-ONES DUPONT PHARMACEUTICALS (US) 2000-10-10 US disclosed