SCHEMBL7052174

SCHEMBL7052174

CCOC(=O)c1cn(CCCN(C=O)OC(C)(C)C)c2cc(CNc3nccn3C(c3ccccc3)(c3ccccc3)c3ccccc3)ccc2c1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 1/20 0.39
CNR1 P21554 8/20 0.34
CNR2 P34972 6/20 0.34
ALDH1A1 P00352 2/20 0.33
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
TDP1 Q9NUW8 1/20 0.32
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
PIM1 P11309 1/20 0.31
IRAK1 P51617 1/20 0.31
CAMK2B Q13554 1/20 0.31
CAMK2G Q13555 1/20 0.31
CAMK2D Q13557 1/20 0.31
PIM3 Q86V86 1/20 0.31
GNRHR P30968 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5663495 0.94 P2RX3 (0.38) P2RX3CNR1CNR2ALDH1A1TDP1
SCHEMBL5663451 0.93 CNR1 (0.35) CNR1CNR2ITGB3ITGAV
SCHEMBL4654781 0.85 P2RX3 (0.40) P2RX3CNR1CNR2ALDH1A1ITGB3
SCHEMBL12372084 0.83 P2RX3 (0.42) P2RX3ALDH1A1TDP1MAPTTSHR
SCHEMBL4654929 0.77 CAMK2D (0.37) CNR1CNR2ITGB3ITGAVCAMK2D
SCHEMBL5662320 0.76 KMT2A (0.41) P2RX3CNR1CNR2ALDH1A1TDP1
SCHEMBL5665792 0.76 LMNA (0.52) P2RX3CNR1CNR2ALDH1A1TDP1
SCHEMBL5779683 0.76 S1PR1 (0.36) P2RX3CNR1ALDH1A1
SCHEMBL5663750 0.75 KMT2A (0.44) P2RX3CNR1CNR2ALDH1A1TDP1
SCHEMBL4388255 0.74 S1PR1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1307226-A2 VITRONECTIN RECEPTOR ANTAGONIST PHARMACEUTICALS Bristol-Myers Squibb Pharma Company (US) 2003-05-07 EP disclosed
WO-2001097848-A2 VITRONECTIN RECEPTOR ANTAGONIST PHARMACEUTICALS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2001-12-27 WO disclosed