SCHEMBL5779711

SCHEMBL5779711

CC1(C)C(=O)C(C)(C)c2cc(C(O)CN3CCN(c4snc5ccccc45)CC3)ccc21

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.39
DRD2 P14416 1/20 0.39
HTR2A P28223 1/20 0.39
HTR7 P34969 1/20 0.38
ALDH1A1 P00352 1/20 0.37
ATM Q13315 1/20 0.37
ADRA1D P25100 10/20 0.36
ADRA1A P35348 10/20 0.36
ADRA1B P35368 10/20 0.36
ADRB2 P07550 9/20 0.36
ADRB1 P08588 9/20 0.36
ADRB3 P13945 9/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
IGF1R P08069 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5738728 0.91 MEN1 (0.39) HTR1AKMT2AMEN1
SCHEMBL5737988 0.89 HTR1A (0.30) HTR1ADRD2HTR2A
SCHEMBL6400409 0.83
SCHEMBL5739938 0.80 MAPT (0.42) ALDH1A1
SCHEMBL5776547 0.79 POLB (0.39) HTR1A
SCHEMBL6400812 0.78 HTR2A (0.47) HTR1ADRD2HTR2AHTR7
SCHEMBL6400851 0.75
SCHEMBL5738711 0.73 MEN1 (0.39) HTR1AKMT2AMEN1
SCHEMBL6399272 0.72 DRD2 (0.44) DRD2HTR2A
SCHEMBL5738525 0.72 HTR1A (0.44) HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1697334-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA Warner-Lambert Company LLC (US) 2006-09-06 EP disclosed
WO-2005056540-A1 HETEROCYCLIC SUBSTITUTED INDANE DERIVATIVES AND RELATED COMPOUNDS FOR THE TREATMENT OF SCHIZOPHRENIA WARNER-LAMBERT COMPANY LLC (US) 2005-06-23 WO disclosed