SCHEMBL5779902

SCHEMBL5779902

COC(=O)[C@H](Cc1ccc(I)cc1)NCCCS(=O)(=O)O.O=S(=O)(O)CCC[n+]1ccc(-c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.40
HDAC6 Q9UBN7 4/20 0.40
SIGMAR1 Q99720 2/20 0.39
CA12 O43570 2/20 0.38
CA7 P43166 2/20 0.38
CA9 Q16790 2/20 0.38
CA14 Q9ULX7 2/20 0.38
CA2 P00918 1/20 0.38
POLB P06746 2/20 0.37
TSHR P16473 1/20 0.36
MDM4 O15151 1/20 0.36
MDM2 Q00987 1/20 0.36
ATM Q13315 1/20 0.36
CDK2 P24941 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13330263 0.87 PTPRB (0.40) HDAC1HDAC6SIGMAR1CA12CA7
SCHEMBL929646 0.87 PTPRB (0.40) HDAC1HDAC6SIGMAR1CA12CA7
SCHEMBL14285091 0.82 CA12 (0.52) CA12CA7CA9CA14CA2
SCHEMBL12226563 0.77 ATM (0.47) HDAC1HDAC6CA12CA7CA9
SCHEMBL14099736 0.76 LNPEP (0.42) HDAC1HDAC6CA12CA7CA9
SCHEMBL12226761 0.76 CA12 (0.52) HDAC1HDAC6CA12CA7CA9
SCHEMBL10231021 0.74 ALDH1A1 (0.47) HDAC1HDAC6CA12CA7CA9
SCHEMBL16472042 0.74 ATM (0.46) HDAC1HDAC6CA12CA7CA9
SCHEMBL352625 0.74 MMP8 (0.47) CA12CA7CA9CA14CA2
SCHEMBL352624 0.74 MMP8 (0.47) CA12CA7CA9CA14CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1646659-A2 IMPROVED PHARMACEUTICAL DRUG CANDIDATES AND METHODS FOR PREPARATION THEREOF Neurochem (International) Limited (CH) 2006-04-19 EP disclosed
WO-2004113391-A2 IMPROVED PHARMACEUTICAL DRUG CANDIDATES AND METHODS FOR PREPARATION THEREOF NEUROCHEM (INTERNATIONAL) LIMITED (CH) 2004-12-29 WO disclosed