SCHEMBL5780375

SCHEMBL5780375

FC(F)(F)c1ccc(COCc2ccc(Cl)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 4/20 0.57
KMT2A Q03164 1/20 0.49
PPARG P37231 1/20 0.48
PPARA Q07869 1/20 0.48
MAOB P27338 4/20 0.47
AGXT P21549 2/20 0.47
P2RX3 P56373 1/20 0.46
KCNH2 Q12809 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
SLC6A4 P31645 1/20 0.46
CNR2 P34972 1/20 0.45
OPRL1 P41146 1/20 0.44
CNR1 P21554 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
TACR1 P25103 1/20 0.42
CYP19A1 P11511 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL492736 0.89 IDO1 (0.68) IDO1KMT2AMAOBTAAR1TACR1
Hydroxyamine SCHEMBL8924228 0.83 IDO1 (0.67) IDO1KMT2AMAOBTAAR1
SCHEMBL5782964 0.83 GRIN2B (0.52) IDO1MAOBAGXTTACR1
SCHEMBL4995796 0.82 IDO1 (0.64) IDO1KMT2AMAOBAGXTSLC6A4
SCHEMBL8076361 0.82 IDO1 (0.59) IDO1KMT2AMAOBTAAR1TACR1
SCHEMBL11926053 0.81 P2RX3 (0.50) IDO1PPARGPPARAMAOBP2RX3
SCHEMBL8995755 0.80 IDO1 (0.61) IDO1KMT2AMAOBAGXTSLC6A4
SCHEMBL668193 0.80 IDO1 (0.57) IDO1KMT2AMAOBTAAR1TACR1
SCHEMBL196588 0.80 CYP19A1 (0.55) KMT2AP2RX3CYP19A1
SCHEMBL28777340 0.80 CYP19A1 (0.55) KMT2AP2RX3CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1620086-A1 COMPOUNDS THAT MODULATE PPAR ACTIVITY AND METHODS OF PREPARATION Warner-Lambert Company LLC (US) 2006-02-01 EP disclosed
WO-2004091604-A1 COMPOUNDS THAT MODULATE PPAR ACTIVITY AND METHODS OF PREPARATION WARNER-LAMBERT COMPANY LLC (US) 2004-10-28 WO disclosed