SCHEMBL5780773

SCHEMBL5780773

COc1ccc2nccc(N3CCN(CC(C)N)CC3)c2n1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.38
CYP8B1 Q9UNU6 1/20 0.37
SLC2A1 P11166 4/20 0.37
EHMT2 Q96KQ7 1/20 0.35
EHMT1 Q9H9B1 1/20 0.35
OGA O60502 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4069340 0.84 KCNH2 (0.42) KCNH2EHMT2EHMT1
SCHEMBL16986089 0.84 KCNH2 (0.40) KCNH2SLC2A1
SCHEMBL1223381 0.84 KCNH2 (0.40) KCNH2SLC2A1
SCHEMBL16986085 0.84 KCNH2 (0.40) KCNH2SLC2A1
SCHEMBL4068487 0.81 EHMT2 (0.41) KCNH2CYP8B1EHMT2EHMT1
SCHEMBL4069756 0.80 KCNH2 (0.41) KCNH2EHMT2EHMT1
Hydrochloric Acid SCHEMBL4069318 0.79 EHMT2 (0.46) KCNH2CYP8B1EHMT2EHMT1
SCHEMBL4068537 0.78 CYP8B1 (0.41) KCNH2CYP8B1EHMT2EHMT1
SCHEMBL1222834 0.77 CYP2C19 (0.46) KCNH2CYP8B1
SCHEMBL1222623 0.77 NCF1 (0.57) CYP8B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1605938-A4 ANTIBACTERIAL AGENTS GLAXO GROUP LTD (GB) 2006-11-22 EP disclosed
EP-1605938-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2005-12-21 EP disclosed
WO-2004087145-A2 ANTIBACTERIAL AGENTS GLAXO GROUP LIMITED (GB) 2004-10-14 WO disclosed