Cyclopentanamine

Cyclopentanamine

SCHEMBL578697

NC1CCCC1.O=C(O)O

nearest known ligand 0.62

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Cyclopentanamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MMP8 P22894 2/20 0.38
MMP1 P03956 1/20 0.38
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
GABRR1 P24046 1/20 0.36
MMP2 P08253 1/20 0.36
EPHX1 P07099 3/20 0.36
LMNA P02545 1/20 0.35
OAT P04181 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cyclohexylamine SCHEMBL578785 0.97 CES2 (0.43) THRBALDH1A1MMP8MMP1CES2
Cyclooctanamine SCHEMBL11193013 0.97 CES2 (0.43) THRBALDH1A1MMP8MMP1CES2
Cycloheptanamine SCHEMBL720218 0.97 CES2 (0.43) THRBALDH1A1MMP8MMP1CES2
Cyclohexylamine SCHEMBL974340 0.97 CES2 (0.43) THRBALDH1A1MMP8MMP1CES2
Cyclohexylamine SCHEMBL27712727 0.91 ALDH1A1 (0.39) ALDH1A1MMP8MMP1CES2CES1
Cyclopentanamine SCHEMBL3875980 0.90 ACHE (0.44) THRBMEN1KMT2AALDH1A1MMP8
Bicarbonate SCHEMBL578685 0.90
Bicarbonate SCHEMBL7136153 0.89 GABRR1 (0.42) GABRR1LMNAOAT
Bicarbonate SCHEMBL7136582 0.89 GABRR1 (0.42) GABRR1LMNAOAT
Bicarbonate SCHEMBL1702507 0.89

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 56 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3169403-B9 ORAL PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY BOWEL DISEASES PROTAGONIST THERAPEUTICS INC (US) 2024-07-03 EP claimed
EP-3169403-B1 ORAL PEPTIDE INHIBITORS OF INTERLEUKIN-23 RECEPTOR AND THEIR USE TO TREAT INFLAMMATORY BOWEL DISEASES PROTAGONIST THERAPEUTICS INC (US) 2024-02-14 EP claimed
EP-1765408-B1 POLYPEPTIDE PROTRACTING TAGS COMPRISING A TETRAZOLE MOIETY NOVO NORDISK AS (DK) 2015-12-09 EP claimed
EP-2289560-B1 POLYPEPTIDE PROTRACTING TAGS COMPRISING A TETRAZOLE MOIETY NOVO NORDISK AS (DK) 2015-04-22 EP claimed
EP-2462147-B1 CONFORMATIONALLY CONSTRAINED, FULLY SYNTHETIC MACROCYCLIC COMPOUNDS POLYPHOR AG (CH) 2014-11-12 EP claimed
EP-2516009-B1 SUBSTITUTED ISOQUINOLINONES AND QUINAZOLINONES NOVARTIS AG (CH) 2014-09-24 EP claimed
EP-2231701-B1 PEPTIDOMIMETICS WITH GLUCAGON ANTAGONISTIC AND GLP-1 AGONISTIC ACTIVITIES CADILA HEALTHCARE LTD (IN) 2012-04-18 EP claimed
EP-1883451-B9 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON INC (CA) 2011-02-09 EP claimed
EP-1883451-B1 SUBSTITUTED INDOLE COMPOUNDS HAVING NOS INHIBITORY ACTIVITY NEURAXON INC (CA) 2010-11-24 EP claimed
EP-1006122-B1 PHENETHYLAMINE DERIVATIVES CHUGAI PHARMACEUTICAL CO LTD (JP) 2008-12-03 EP claimed
EP-1257575-B1 RADIOLABELED VASOACTIVE INTESTINAL PEPTIDE ANALOGS FOR DIAGNOSIS AND RADIOTHERAPY DABUR RES FOUNDATION (IN) 2007-02-28 EP claimed
EP-1337551-B1 SUBSTANCE P ANALOGS FOR THE TREATMENT OF CANCER DABUR PHARMA LTD (IN) 2007-01-03 EP claimed
EP-1165099-B1 ANGIOTENSIN II AND ANALOGS THEREOF FOR LIMITING SCAR AND ADHESION FORMATION UNIV SOUTHERN CALIFORNIA (US) 2006-08-09 EP claimed
EP-1257576-B1 VASOACTIVE INTESTINAL PEPTIDE ANALOGS DABUR RES FOUNDATION (IN) 2004-09-15 EP claimed
EP-0606881-B1 Cyclic pentapeptides having a beta-turn and a gamma-turn TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-05-12 EP claimed
EP-0245961-B1 ACID GAS SCRUBBING COMPOSITION AND PROCESS EXXON RESEARCH AND ENGINEERING COMPANY (US) 1991-04-03 EP claimed
EP-2708569-B1 TRANSPARENT POLYAMIDE-IMIDES EMS PATENT AG (CH) 2018-05-23 EP disclosed
EP-2708569-A1 Transparent polyamidimide EMS-PATENT AG (CH) 2014-03-19 EP disclosed
EP-0284942-A2 Amino-acid derivatives MERCK PATENT GmbH (DE) 1988-10-05 EP disclosed
EP-0068373-A1 Schiff bases of aminocycloalcanecarboxylic esters, preparation thereof and use thereof as intermediate products BASF Aktiengesellschaft (DE) 1983-01-05 EP disclosed