SCHEMBL5790711

SCHEMBL5790711

CC(C)(C)OC(=O)N1CCCC(CNC(=O)c2cc(-c3ccc(Cl)cc3)ccc2N)C1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.54
KAT7 O95251 1/20 0.46
KAT8 Q9H7Z6 1/20 0.46
USP30 Q70CQ3 1/20 0.45
KMT2A Q03164 3/20 0.45
MEN1 O00255 1/20 0.45
KAT6A Q92794 1/20 0.45
KAT5 Q92993 1/20 0.45
ALDH1A1 P00352 3/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC2 Q92769 1/20 0.44
KDM4E B2RXH2 1/20 0.44
PKM P14618 1/20 0.44
CNR1 P21554 1/20 0.44
CNR2 P34972 1/20 0.44
CYP2C9 P11712 1/20 0.43
IRAK1 P51617 1/20 0.42
KDM1A O60341 1/20 0.42
SCN9A Q15858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791461 0.86 KMT2A (0.49) KMT2AMEN1ALDH1A1KDM4E
SCHEMBL5791116 0.85 ACKR3 (0.55) ACKR3KAT7KAT8USP30KMT2A
SCHEMBL5792816 0.82 CCR2 (0.47) KMT2AMEN1ALDH1A1
SCHEMBL3765452 0.77 ACKR3 (0.60) ACKR3USP30KMT2AMEN1ALDH1A1
SCHEMBL13056746 0.77 ACKR3 (0.60) ACKR3USP30KMT2AMEN1ALDH1A1
SCHEMBL3448188 0.77 KDM4E (0.69) ACKR3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL3448190 0.77 KDM4E (0.69) ACKR3KMT2AMEN1ALDH1A1KDM4E
SCHEMBL2070349 0.77 PPARA (0.61) ACKR3CNR1CNR2CYP2C9
SCHEMBL4847812 0.76 CCR2 (0.57) KMT2AMEN1KDM4EPKM
SCHEMBL2069204 0.75 CHEK2 (0.59) ACKR3KAT7KAT8KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006012577-A2 QUINAZOLINONE DERIVATIVES USEFUL FOR THE REGULATION OF GLUCOSE HOMEOSTASIS AND FOOD INTAKE BAYER PHARMACEUTICALS CORPORATION (US) 2006-02-02 WO disclosed