SCHEMBL5790846

SCHEMBL5790846

COc1nc(=O)c2c(C)cccc2n1OC

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.40
ELANE P08246 5/20 0.39
P2RX7 Q99572 2/20 0.33
PARP1 P09874 1/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 3/20 0.33
KMT2A Q03164 3/20 0.33
LMNA P02545 2/20 0.33
HIF1A Q16665 2/20 0.33
PDE2A O00408 1/20 0.33
PDE6D O43924 1/20 0.33
PDE6A P16499 1/20 0.33
PDE6G P18545 1/20 0.33
PDE4A P27815 1/20 0.33
PDE6B P35913 1/20 0.33
PDE6C P51160 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE6H Q13956 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3974206 0.68 SMN1; SMN2 (0.44) SMN1; SMN2ALDH1A1KDM4ELMNAPDE2A
SCHEMBL29150251 0.64 ELANE (0.49) SMN1; SMN2ELANEALDH1A1KDM4EKMT2A
SCHEMBL11076238 0.61 TDP2 (0.45) SMN1; SMN2ALDH1A1KDM4EKMT2ATP53
SCHEMBL10439112 0.60 SMN1; SMN2 (0.47) SMN1; SMN2ELANEALDH1A1KDM4EKMT2A
SCHEMBL149479 0.60 ALDH1A1 (0.68) SMN1; SMN2ALDH1A1KDM4EKMT2ALMNA
SCHEMBL5775044 0.59 ALDH1A1 (0.38) SMN1; SMN2ELANEPARP1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL31716024 0.59 ALDH1A1 (0.66) SMN1; SMN2ALDH1A1KDM4EKMT2ALMNA
Hydrochloric Acid SCHEMBL15709616 0.59 ALDH1A1 (0.66) SMN1; SMN2ALDH1A1KDM4EKMT2ALMNA
SCHEMBL18317487 0.59 SMN1; SMN2 (0.60) SMN1; SMN2ALDH1A1KDM4EKMT2ABACE1
SCHEMBL366928 0.58 IDO1 (0.45) SMN1; SMN2ALDH1A1KMT2ALMNAHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1644369-A2 ARYLAMINE-SUBSTITUTED QUINAZOLINONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-04-12 EP disclosed
WO-2005005395-A2 ARYLAMINE-SUBSTITUTED QUINAZOLINONE COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-01-20 WO disclosed