SCHEMBL5790636

SCHEMBL5790636

CC(C)(C)CN(NC(=O)c1ccc(F)c(F)c1)c1ccnc(C#N)n1

nearest known ligand 0.44

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSK P43235 10/20 0.44
KCNQ3 O43525 4/20 0.40
KCNQ2 O43526 4/20 0.40
CTSB P07858 2/20 0.38
CTSS P25774 2/20 0.38
CTSC P53634 2/20 0.38
CTSL P07711 1/20 0.38
FGFR4 P22455 1/20 0.37
MCHR1 Q99705 1/20 0.34
KCNQ5 Q9NR82 1/20 0.34
S1PR3 Q99500 2/20 0.34
AR P10275 1/20 0.34
GPR4 P46093 1/20 0.34
S1PR1 P21453 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791503 0.89 CTSK (0.47) CTSKCTSBCTSSCTSCCTSL
SCHEMBL8271448 0.87 CTSK (0.46) CTSKCTSLFGFR4AR
SCHEMBL8268844 0.83 CTSK (0.45) CTSKCTSBCTSSCTSCCTSL
SCHEMBL8270467 0.83 CTSK (0.48) CTSKCTSBCTSSCTSCCTSL
SCHEMBL5791966 0.82 CTSK (0.45) CTSKCTSSCTSLFGFR4
SCHEMBL8271447 0.82 CTSK (0.43) CTSKFGFR4
SCHEMBL5792274 0.82 CTSK (0.43) CTSKCTSSMCHR1
SCHEMBL8270779 0.79 CTSK (0.40) CTSKCTSBCTSSCTSCCTSL
SCHEMBL8270485 0.78 CTSK (0.37) CTSKCTSBCTSSCTSCCTSL
SCHEMBL5791397 0.78 CTSK (0.48) CTSKCTSBCTSSCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed