SCHEMBL5791897

SCHEMBL5791897

CC(C)CN(c1ccnc(C#N)n1)N(CCCCCN1C(=O)c2ccccc2C1=O)C(=O)O

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 0.41
ACHE P22303 7/20 0.41
BCHE P06276 2/20 0.40
CTSK P43235 1/20 0.37
KDM4E B2RXH2 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791906 0.99 MAOB (0.40) MAOBACHEBCHECTSK
SCHEMBL5792592 0.96 MAOB (0.39) MAOBACHEBCHECTSK
SCHEMBL8270740 0.89 MAOB (0.35) MAOBACHEBCHECTSK
SCHEMBL8270736 0.88 CTSK (0.35) MAOBACHEBCHECTSK
SCHEMBL8270739 0.85 CTSK (0.35) MAOBACHEBCHECTSK
SCHEMBL5791444 0.83 CTSK (0.40) CTSK
SCHEMBL5794663 0.82 CTSK (0.39) CTSKKDM4E
SCHEMBL5791034 0.80 CTSK (0.42) CTSKKDM4E
SCHEMBL5794549 0.79 CTSK (0.41) CTSK
SCHEMBL5795031 0.76 CTSK (0.35) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed