SCHEMBL579203

SCHEMBL579203

O=C1NC(=O)c2c(C=S)cccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.46
PARP1 P09874 5/20 0.44
KDM4E B2RXH2 5/20 0.44
ALDH1A1 P00352 4/20 0.44
HSD17B10 Q99714 3/20 0.44
HPGD P15428 2/20 0.44
GAA P10253 1/20 0.44
CASP3 P42574 4/20 0.41
CASP7 P55210 2/20 0.41
CASP2 P42575 1/20 0.41
CASP6 P55212 1/20 0.41
CASP8 Q14790 1/20 0.41
POLB P06746 3/20 0.37
NPSR1 Q6W5P4 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
RGS12 O14924 1/20 0.37
USP2 O75604 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31229225 0.82 GSK3B (0.48) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL1627401 0.82 GSK3B (0.48) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL626418 0.81 GSK3B (0.46) GSK3BPARP1KDM4EALDH1A1HSD17B10
Iodide SCHEMBL2495412 0.79 GSK3B (0.45) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL8577337 0.78 KDM4E (0.45) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL16754925 0.77 GSK3B (0.62) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL28735098 0.75 GSK3B (0.41) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL7552794 0.74 KDM4E (0.42) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL7693227 0.74 KDM4E (0.42) GSK3BPARP1KDM4EALDH1A1HSD17B10
SCHEMBL6510808 0.74 GSK3B (0.52) GSK3BPARP1KDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417122-A1 INDOLE DERIVATIVES AND METHODS FOR ANTIVIRAL TREATMENT PTC Therapeutics, Inc. (US) 2012-02-15 EP disclosed
WO-2010117932-A1 INDOLE DERIVATIVES AND METHODS FOR ANTIVIRAL TREATMENT SCHERING CORPORATION (US) 2010-10-14 WO disclosed