SCHEMBL5793583

SCHEMBL5793583

C[C@H](N)C(=O)N[C@H]1CC(c2ccccc2)=CCN(C)C1=O

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
XIAP P98170 15/20 0.47
TAAR1 Q96RJ0 1/20 0.39
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
MME P08473 1/20 0.35
ACE P12821 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5793580 0.81 KDM1A (0.41) XIAPMEN1KMT2AKCNH2HRH3
SCHEMBL5794399 0.81 XIAP (0.47) XIAPTAAR1HDAC1HDAC2HDAC8
SCHEMBL5794437 0.79 XIAP (0.43) XIAPTAAR1KCNH2
SCHEMBL5793470 0.79 XIAP (0.43) XIAPTAAR1KCNH2
SCHEMBL5793607 0.78 TAAR1 (0.40) XIAPTAAR1HDAC1HDAC2HDAC8
SCHEMBL4837323 0.77 PSEN1 (0.51) XIAP
SCHEMBL4841337 0.77 PSEN1 (0.55)
Hydrochloric Acid SCHEMBL25345659 0.75 XIAP (0.53) XIAPMMEACE
Hydrochloric Acid SCHEMBL25345671 0.75 XIAP (0.53) XIAPMMEACE
Hydrochloric Acid SCHEMBL25345665 0.75 XIAP (0.53) XIAPMMEACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636196-A1 NOVEL LACTAMS AND USES THEREOF AstraZeneca AB (SE) 2006-03-22 EP claimed
WO-2004080983-A1 NOVEL LACTAMS AND USES THEREOF ASTRAZENECA AB (SE) 2004-09-23 WO claimed
EP-1636196-A1 NOVEL LACTAMS AND USES THEREOF AstraZeneca AB (SE) 2006-03-22 EP disclosed
WO-2004080983-A1 NOVEL LACTAMS AND USES THEREOF ASTRAZENECA AB (SE) 2004-09-23 WO disclosed