Pyrene

Pyrene

SCHEMBL5793586

c1cc2ccc3cccc4ccc(c1)c2c34.c1ccc2c(c1)Cc1ccccc1-2.c1ccc2c(c1)ccc1ccccc12

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 7/20 0.56
CYP3A4 P08684 3/20 0.56
ALDH1A1 P00352 10/20 0.48
HSD17B10 Q99714 10/20 0.48
CYP2A6 P11509 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
CYP1A2 P05177 4/20 0.47
MAOA P21397 2/20 0.47
ERBB2 P04626 1/20 0.47
FYN P06241 1/20 0.47
ACHE P22303 1/20 0.47
AHR P35869 1/20 0.47
HPGD P15428 7/20 0.46
THRB P10828 1/20 0.46
KDM4E B2RXH2 4/20 0.46
HPRT1 P00492 1/20 0.44
CYP1B1 Q16678 2/20 0.44
CYP1A1 P04798 1/20 0.44
MAPK1 P28482 4/20 0.43
L3MBTL1 Q9Y468 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenanthrene SCHEMBL21219119 0.92 TSHR (0.57) TSHRCYP3A4ALDH1A1HSD17B10CYP2A6
Pyrene SCHEMBL2125072 0.92 TSHR (0.65) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2
Pyrene SCHEMBL1133715 0.91 CYP1A2 (0.49) TSHRCYP3A4ALDH1A1HSD17B10CYP2A6
Benzo[E]Pyrene SCHEMBL28074705 0.88 ALDH1A1 (0.64) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2
Fluorene SCHEMBL7752293 0.88 TSHR (0.54) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2
Fluorene SCHEMBL28556215 0.88 TSHR (0.54) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2
Fluorene SCHEMBL28714196 0.85 MAOA (0.48) TSHRCYP3A4ALDH1A1HSD17B10CYP2A6
Phenanthrene SCHEMBL5161188 0.84 TSHR (0.48) TSHRCYP3A4ALDH1A1HSD17B10CYP2A6
Fluorene SCHEMBL28064647 0.83 TSHR (0.56) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2
SCHEMBL29573523 0.81 TSHR (0.62) TSHRCYP3A4ALDH1A1HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006042187-A2 SIMULTANEOUS SEQUENCE ANALYSIS OF AMINO- AND CARBOXY- TERMINI UNIVERSITY OF VIRGINIA PATENT FOUNDATION (US) 2006-04-20 WO disclosed