SCHEMBL5794096

SCHEMBL5794096

C[C@H](N)C(=O)N[C@H]1CC(c2ccccc2)=C[C@@H](c2ccccc2)NC1=O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
XIAP P98170 11/20 0.39
TAAR1 Q96RJ0 1/20 0.38
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
CTSK P43235 3/20 0.33
CTSL P07711 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5794668 1.00 XIAP (0.39) XIAPTAAR1HDAC1HDAC2HDAC8
SCHEMBL5794093 0.82 KDM1A (0.45)
SCHEMBL5794664 0.82 KDM1A (0.45)
SCHEMBL4843190 0.78 PSEN1 (0.44)
SCHEMBL4839952 0.78 PSEN1 (0.44)
SCHEMBL5794458 0.78 XIAP (0.39) XIAPTAAR1
SCHEMBL5793607 0.78 TAAR1 (0.40) XIAPTAAR1HDAC1HDAC2HDAC8
SCHEMBL4842242 0.78 PSEN1 (0.49)
SCHEMBL4842158 0.78 PSEN1 (0.49)
SCHEMBL5794437 0.77 XIAP (0.43) XIAPTAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1636196-A1 NOVEL LACTAMS AND USES THEREOF AstraZeneca AB (SE) 2006-03-22 EP disclosed
WO-2004080983-A1 NOVEL LACTAMS AND USES THEREOF ASTRAZENECA AB (SE) 2004-09-23 WO disclosed