SCHEMBL5794299

SCHEMBL5794299

CCN1CCC[C@H](Cn2c(C(C)C)nc3ccc(Br)cc3c2=O)C1

nearest known ligand 0.57

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 7/20 0.57
HTR2C P28335 1/20 0.53
CACNA2D1 P54289 11/20 0.50
OPRM1 P35372 1/20 0.48
GHSR Q92847 4/20 0.45
KCNH2 Q12809 2/20 0.43
CYP3A4 P08684 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5791009 0.87 CYP2D6 (0.74) CYP2D6CACNA2D1GHSRKCNH2CYP3A4
SCHEMBL5792111 0.86 CYP2D6 (0.56) CYP2D6CACNA2D1OPRM1GHSRKCNH2
SCHEMBL5793556 0.86 CYP2D6 (0.56) CYP2D6CACNA2D1OPRM1GHSRKCNH2
SCHEMBL5793560 0.86 CYP2D6 (0.56) CYP2D6CACNA2D1OPRM1GHSRKCNH2
SCHEMBL5823927 0.83 CYP2D6 (0.80) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5791006 0.81 CYP2D6 (0.67) CYP2D6CACNA2D1GHSRKCNH2CYP3A4
SCHEMBL5792392 0.81 CYP2D6 (0.51) CYP2D6CACNA2D1OPRM1GHSRKCNH2
SCHEMBL5794769 0.81 CYP2D6 (0.62) CYP2D6HTR2CGHSRKCNH2CYP3A4
SCHEMBL5790809 0.77 GHSR (0.58) CYP2D6CACNA2D1GHSRKCNH2CYP3A4
SCHEMBL5791730 0.77 GHSR (0.73) CYP2D6GHSRKCNH2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006012577-A2 QUINAZOLINONE DERIVATIVES USEFUL FOR THE REGULATION OF GLUCOSE HOMEOSTASIS AND FOOD INTAKE BAYER PHARMACEUTICALS CORPORATION (US) 2006-02-02 WO disclosed