SCHEMBL5795015

SCHEMBL5795015

CCCN1CCN(Cc2ccc(C(=O)N(NCC(C)(C)C)c3ccnc(C#N)n3)cc2)CC1

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSK P43235 13/20 0.44
CTSL P07711 3/20 0.44
CTSS P25774 3/20 0.44
CTSB P07858 1/20 0.40
GPR4 P46093 2/20 0.38
JAK2 O60674 2/20 0.36
JAK3 P52333 2/20 0.36
TBK1 Q9UHD2 2/20 0.36
IKBKE Q14164 1/20 0.36
HDAC6 Q9UBN7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5793222 0.89 CTSK (0.41) CTSKCTSLCTSSCTSBGPR4
Trifluoroacetic Acid SCHEMBL5795046 0.86 HRH4 (0.41) CTSKCTSLCTSSCTSB
SCHEMBL8270035 0.81 CTSK (0.51) CTSKCTSLCTSSCTSBGPR4
Trifluoroacetic Acid SCHEMBL5794574 0.78 CTSK (0.48) CTSKCTSLCTSSCTSBGPR4
Trifluoroacetic Acid SCHEMBL5804566 0.78 CTSK (0.46) CTSKCTSLCTSSCTSBGPR4
SCHEMBL8270525 0.76 CTSK (0.63) CTSKCTSLCTSSCTSBGPR4
SCHEMBL5529854 0.74 CTSL (0.44) CTSKCTSLCTSSCTSBJAK2
SCHEMBL5500170 0.74 CTSK (0.58) CTSKCTSLCTSSCTSBGPR4
Trifluoroacetic Acid SCHEMBL5791240 0.74 CTSK (0.57) CTSKCTSLCTSSCTSBGPR4
SCHEMBL5522122 0.72 CTSK (0.41) CTSKCTSLCTSSCTSBTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO claimed