SCHEMBL5797428

SCHEMBL5797428

COc1ccc2nc(NCC(C)=Cc3ccc(C(=O)NO)cc3)sc2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCD O00767 13/20 0.58
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
MEN1 O00255 2/20 0.58
KMT2A Q03164 2/20 0.58
TOP2A P11388 3/20 0.56
CYP1A2 P05177 1/20 0.53
CYP3A4 P08684 1/20 0.53
CYP2C19 P33261 1/20 0.53
HTT P42858 1/20 0.53
DYRK1A Q13627 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
KDM4E B2RXH2 1/20 0.52
ALDH1A1 P00352 1/20 0.52
GAA P10253 1/20 0.52
MAPT P10636 1/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
HDAC1 Q13547 1/20 0.51
CASP2 P42575 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795590 0.90 TOP2A (0.58) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5799660 0.90 TOP2A (0.58) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5807692 0.83 KMT2A (0.55) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5799236 0.80 SCD (0.47) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5809983 0.79 SCD (0.46) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5809988 0.79 SCD (0.46) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5811548 0.79 HDAC6 (0.63) NPC1RAB9AALDH1A1HPGDHDAC1
SCHEMBL5811555 0.79 HDAC6 (0.63) NPC1RAB9AALDH1A1HPGDHDAC1
SCHEMBL5653631 0.76 NPC1 (0.64) SCDNPC1RAB9AMEN1KMT2A
SCHEMBL5797063 0.76 KMT2A (0.55) SCDNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO claimed
WO-2006025683-A1 ARYLAMINOMETHYL PROPENYL BENZHYDROXYAMID DERIVATIVES WITH INHIBITORY ACTIVITY AGAINST HISTONE DEACETYLASE AND METHOD FOR THE PREPARATION THEREOF KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2006-03-09 WO disclosed