SCHEMBL5798044

SCHEMBL5798044

Cc1c(C(C(=O)O)C2CCCC2)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(OC(F)(F)F)cc1.Cc1c(CC(=O)Nc2c(C)n(C(=O)c3ccc(OC(F)(F)F)cc3)c3cc(F)c(O)c(F)c23)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(OC(F)(F)F)cc1.Cc1c(CC(=O)O)c2c(F)c(O)c(F)cc2n1C(=O)c1ccc(OC(F)(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 8/20 0.37
AKR1C2 P52895 8/20 0.37
PTGS2 P35354 8/20 0.36
MAPT P10636 4/20 0.36
TP53 P04637 1/20 0.36
ABCB1 P08183 2/20 0.36
PTGS1 P23219 2/20 0.36
AKR1C4 P17516 2/20 0.36
AKR1C1 Q04828 2/20 0.36
KMT2A Q03164 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
PPARG P37231 2/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
PTGES O14684 1/20 0.36
ABCC3 O15438 1/20 0.36
ABCC4 O15439 1/20 0.36
ABCB11 O95342 1/20 0.36
MT-CO2 P00403 1/20 0.36
LMNA P02545 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6426016 0.88 HSD11B1 (0.38) PTGS2PPARG
SCHEMBL6423536 0.86 HSD11B1 (0.38) PPARGPTGDR2
SCHEMBL5554589 0.81 AKR1C3 (0.53) AKR1C3AKR1C2PTGS2MAPTABCB1
SCHEMBL5554131 0.78 PTGS2 (0.46) AKR1C3AKR1C2PTGS2
SCHEMBL5558197 0.78 PTGS2 (0.48) AKR1C3AKR1C2PTGS2PPARG
SCHEMBL5553844 0.77 PTGS2 (0.49) AKR1C3AKR1C2PTGS2ABCB1PTGS1
SCHEMBL6423593 0.77 HSD11B1 (0.39) AKR1C3AKR1C2PTGS2PPARG
SCHEMBL6425845 0.77 PTGS2 (0.38) PTGS2PPARGKDM4EPTGDR2
SCHEMBL6427040 0.77 PTGS2 (0.53) AKR1C3AKR1C2PTGS2MAPTTP53
SCHEMBL6423869 0.77 AKR1C3 (0.39) AKR1C3AKR1C2PTGS2ABCB1PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed