SCHEMBL5798252

SCHEMBL5798252

CC(=O)CCC(Br)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LCK P06239 1/20 0.50
PPARD Q03181 1/20 0.50
ZDHHC20 Q5W0Z9 1/20 0.50
ZDHHC2 Q9UIJ5 1/20 0.50
ALDH1A1 P00352 5/20 0.46
TSHR P16473 1/20 0.46
LMNA P02545 1/20 0.42
SLC15A2 Q16348 1/20 0.42
THRB P10828 1/20 0.36
RECQL P46063 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.35
TRPA1 O75762 1/20 0.35
CHRM1 P11229 1/20 0.33
AKR1A1 P14550 1/20 0.33
CHRM3 P20309 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
ADRA1A P35348 1/20 0.33
HRH1 P35367 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28238506 0.86 LCK (0.57) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL28238495 0.84 LCK (0.61) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL4656310 0.79 TET2 (0.52) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL14893946 0.79 TET2 (0.52) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL16187177 0.79 TET2 (0.52) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL24327258 0.78 ALDH1A1 (0.41) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL2776377 0.78 ALDH1A1 (0.61) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL5965619 0.78 ALDH1A1 (0.61) LCKPPARDZDHHC20ZDHHC2ALDH1A1
SCHEMBL28409342 0.76
SCHEMBL1421677 0.76 ALDH1A1 (0.50) ALDH1A1LMNASLC15A2CYP1A2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106458988-B Heterocycle-butanamide derivatives 默克专利股份公司 2019-12-03 CN disclosed
CN-107709323-A Oxipurinol class compound and its application 广东众生药业股份有限公司 2018-02-16 CN disclosed
EP-1723119-A1 ION CHANNEL MODULATORS Wyeth a Corporation of the State of Delaware (US) 2006-11-22 EP disclosed
WO-2005087747-A1 ION CHANNEL MODULATORS WYETH (US) 2005-09-22 WO disclosed