SCHEMBL5798526

SCHEMBL5798526

O=C(c1cccc(C(F)(F)F)c1)C(Br)c1ccc(=O)[nH]n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.48
CES2 O00748 2/20 0.47
JAK2 O60674 1/20 0.44
NTRK1 P04629 1/20 0.44
RET P07949 1/20 0.44
PDGFRB P09619 1/20 0.44
CDK8 P49336 1/20 0.44
NTRK3 Q16288 1/20 0.44
NTRK2 Q16620 1/20 0.44
AURKB Q96GD4 1/20 0.44
ALDH1A1 P00352 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TLR7 Q9NYK1 3/20 0.40
SRD5A2 P31213 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
MEN1 O00255 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3361277 0.74 CES2 (0.65) CES2ALDH1A1NPSR1SRD5A2MEN1
SCHEMBL6500852 0.73 CES2 (0.56) CES2NPSR1TLR7SRD5A2MEN1
SCHEMBL5797375 0.72 AKR1B1 (0.50) AKR1B1CES2JAK2NTRK1RET
SCHEMBL27627736 0.72 CES2 (0.62) CES2ALDH1A1NPSR1SRD5A2MEN1
Bromide SCHEMBL6282484 0.72 CES2 (0.55) CES2NPSR1TLR7SRD5A2MEN1
SCHEMBL786699 0.71 CES2 (0.61) CES2ALDH1A1NPSR1SRD5A2MEN1
SCHEMBL5796336 0.70 CES2 (0.41) AKR1B1CES2ALDH1A1MEN1KMT2A
SCHEMBL14561095 0.70 CES2 (0.43) CES2ALDH1A1NPSR1TLR7POLB
SCHEMBL27243759 0.69 CES2 (0.71) CES2ALDH1A1NPSR1SRD5A2MEN1
SCHEMBL6601858 0.68 CES2 (0.50) CES2NPSR1TLR7SRD5A2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006038734-A1 PYRIDAZINONE DERIVATIVES CYTOKINES INHIBITORS ASTELLAS PHARMA INC. (JP) 2006-04-13 WO disclosed