SCHEMBL5796336

SCHEMBL5796336

O=C(c1ccccc1F)C(Br)c1ccc(=O)[nH]n1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.41
CES1 P23141 2/20 0.41
AKR1B1 P15121 3/20 0.40
ALDH1A1 P00352 3/20 0.40
HTT P42858 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALOX15 P16050 1/20 0.37
TDP1 Q9NUW8 2/20 0.36
CTNNB1 P35222 1/20 0.36
WNT3A P56704 1/20 0.36
RAB9A P51151 2/20 0.35
NPC1 O15118 1/20 0.35
KMT2A Q03164 3/20 0.35
CYP1A2 P05177 1/20 0.34
GAA P10253 1/20 0.34
MEN1 O00255 2/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4242626 0.84 CES2 (0.43) CES2CES1AKR1B1ALDH1A1HTT
SCHEMBL5797416 0.77 KMT2A (0.43) CES2CES1AKR1B1ALDH1A1HTT
SCHEMBL5798526 0.70 AKR1B1 (0.48) CES2AKR1B1ALDH1A1KMT2AMEN1
SCHEMBL30712874 0.69 CES2 (0.58) CES2CES1ALDH1A1HTTALOX15
SCHEMBL3366577 0.69 CES2 (0.58) CES2CES1ALDH1A1HTTALOX15
SCHEMBL1743417 0.68 CES2 (0.56) CES2CES1ALDH1A1HTTALOX15
SCHEMBL28872295 0.67 ALDH1A1 (0.55) CES2CES1ALDH1A1HTTALOX15
SCHEMBL1155548 0.67 CES2 (0.55) CES2CES1ALDH1A1HTTALOX15
SCHEMBL25310527 0.66 CES2 (0.46) CES2CES1ALDH1A1HTTL3MBTL1
Bromide SCHEMBL25311190 0.65 CES2 (0.45) CES2CES1ALDH1A1HTTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006038734-A1 PYRIDAZINONE DERIVATIVES CYTOKINES INHIBITORS ASTELLAS PHARMA INC. (JP) 2006-04-13 WO disclosed