SCHEMBL5797375

SCHEMBL5797375

O=C(Cc1ccc(=O)[nH]n1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.50
JAK2 O60674 1/20 0.48
NTRK1 P04629 1/20 0.48
RET P07949 1/20 0.48
PDGFRB P09619 1/20 0.48
CDK8 P49336 1/20 0.48
NTRK3 Q16288 1/20 0.48
NTRK2 Q16620 1/20 0.48
AURKB Q96GD4 1/20 0.48
CES2 O00748 1/20 0.48
ALDH1A1 P00352 3/20 0.45
CTNNB1 P35222 1/20 0.43
WNT3A P56704 1/20 0.43
POLB P06746 3/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
SRD5A2 P31213 1/20 0.42
RAB9A P51151 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5795729 0.80 CTNNB1 (0.47) CTNNB1WNT3ALMNAHPGDSMN1; SMN2
SCHEMBL5798675 0.79 CYP1A2 (0.43) AKR1B1ALDH1A1CTNNB1WNT3APOLB
SCHEMBL4245618 0.74 RAB9A (0.51) AKR1B1CES2ALDH1A1CTNNB1WNT3A
SCHEMBL6970291 0.73 CES2 (0.61) CES2ALDH1A1CTNNB1WNT3APOLB
SCHEMBL5799397 0.73 PIM1 (0.45) NTRK1RETPDGFRBCDK8NTRK3
SCHEMBL5798526 0.72 AKR1B1 (0.48) AKR1B1JAK2NTRK1RETPDGFRB
SCHEMBL6133926 0.72 NPSR1 (0.44) AKR1B1CES2ALDH1A1CTNNB1WNT3A
SCHEMBL30758861 0.72 CES2 (0.69) CES2ALDH1A1CTNNB1WNT3APOLB
SCHEMBL423798 0.72 DDR1 (0.59) CES2CTNNB1WNT3ALMNASRD5A2
SCHEMBL28861864 0.72 PTGS1 (0.45) CES2ALDH1A1CTNNB1WNT3APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006038734-A1 PYRIDAZINONE DERIVATIVES CYTOKINES INHIBITORS ASTELLAS PHARMA INC. (JP) 2006-04-13 WO disclosed