SCHEMBL5799245

SCHEMBL5799245

Fc1ccc2c(c1)C(CC1=CNC(=S)[N]1)CC2

nearest known ligand 0.37

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
KDM4C Q9H3R0 1/20 0.33
SLC6A4 P31645 1/20 0.31
KDM2B Q8NHM5 1/20 0.31
IDO1 P14902 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5798616 0.90 ESR1 (0.37) ESR1ESR2SLC6A4KDM2BIDO1
SCHEMBL5802115 0.85 ESR1 (0.37) ESR1ESR2HTR2CSLC6A4KDM2B
SCHEMBL5802150 0.82 HTR6 (0.47) ESR1ESR2IDO1
SCHEMBL5801818 0.78 ESR1 (0.40) ESR1ESR2HTR2AHTR2CKDM4C
SCHEMBL5802349 0.75 SRD5A1 (0.38) ESR1ESR2SLC6A4
SCHEMBL6183415 0.71 DPP4 (0.30)
SCHEMBL1340500 0.71 ESR1 (0.38) ESR1ESR2HTR2AHTR2CKDM4C
SCHEMBL7034308 0.70 ESR1 (0.40) ESR1ESR2HTR2AHTR2CKDM4C
SCHEMBL5800695 0.70 ESR1 (0.37) ESR1ESR2HTR2CSLC6A4
SCHEMBL5801868 0.69 PTGS2 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006036404-A1 4-(SUBSTITUTED CYCLOALKYLMETHYL) IMIDAZOLE-2-THONES, 4-(SUBSTITUTED CYCLOALKENYLMETHYL) IMIDAZOLE-2-THIONES, 4-(SUBSTITUTED CYLOALKYLMETHYL) IMIDAZOL-2-ONES, 4-(SUBSTITUTED CYCLOALKENYLMETHYL) IMIDAZOL-2-ONES AND RELATED COMPOUNDS ALLERGAN, INC. (US) 2006-04-06 WO disclosed